激酶(kinase)是最大且功能最多样的基因家族之一,是重要的药物靶点。激酶是细胞功能的关键调节分子。合研生物提供多种类型激酶靶点,为激酶药物筛选提供基于生化检测及细胞检测服务,还可根据客户药物筛选需求提供多样性选择激酶谱服务。
Target | Assay | Format |
ABL1 | ADP-Glo | 96/384 well |
ABL1(E255K) | ADP-Glo | 96/384 well |
ABL1(T315I) | ADP-Glo | 96/384 well |
ABL1(Y253F) | ADP-Glo | 96/384 well |
ACK | ADP-Glo | 96/384 well |
AKT1 | ADP-Glo | 96/384 well |
AKT2 | ADP-Glo | 96/384 well |
AKT3 | ADP-Glo | 96/384 well |
ALK2 | ADP-Glo | 96/384 well |
ALK4 | ADP-Glo | 96/384 well |
ALK6 | ADP-Glo | 96/384 well |
AMAPK(A1/B1/G2) | ADP-Glo | 96/384 well |
AMPK(A1/B1/G1) | ADP-Glo | 96/384 well |
AMPK(A2/B1/G1) | ADP-Glo | 96/384 well |
ASK1 | ADP-Glo | 96/384 well |
Aurora A | ADP-Glo | 96/384 well |
Aurora B | ADP-Glo | 96/384 well |
AXL | ADP-Glo | 96/384 well |
BRK | ADP-Glo | 96/384 well |
BXM | ADP-Glo | 96/384 well |
Target | Assay | Format |
CAMK1γ |
ADP-Glo |
96/384 well |
CAMK2α |
ADP-Glo |
96/384 well |
CAMK2γ |
ADP-Glo |
96/384 well |
CAMKK1 |
ADP-Glo |
96/384 well |
CDC7/DBF4 |
ADP-Glo |
96/384 well |
CDK2/CyclinA2 |
ADP-Glo |
96/384 well |
CDK2/CyclinE1 |
ADP-Glo |
96/384 well |
CDK3/cyclinE1 |
ADP-Glo |
96/384 well |
CDK5/p25 |
ADP-Glo |
96/384 well |
CDK5/p35 |
ADP-Glo |
96/384 well |
CDK6/CyclinD3 |
ADP-Glo |
96/384 well |
CDK9/Cyclink |
ADP-Glo |
96/384 well |
CHK1 |
ADP-Glo |
96/384 well |
CHK2 |
ADP-Glo |
96/384 well |
CK1a1 |
ADP-Glo |
96/384 well |
CK1γ1 |
ADP-Glo |
96/384 well |
CK1ε |
ADP-Glo |
96/384 well |
CK2α1 |
ADP-Glo |
96/384 well |
c-KIT |
ADP-Glo |
96/384 well |
CLK1 |
ADP-Glo |
96/384 well |
CLK3 |
ADP-Glo |
96/384 well |
c-MER |
ADP-Glo |
96/384 well |
CSK |
ADP-Glo |
96/384 well |
DAPK1 |
ADP-Glo |
96/384 well |
DDR2 |
ADP-Glo |
96/384 well |
DNA-PK |
ADP-Glo |
96/384 well |
DYRK2 | ADP-Glo | 96/384 well |
Target | Assay | Format |
EGFR |
ADP-Glo |
96/384 well |
EGFR(L858R) |
ADP-Glo |
96/384 well |
EGFR(L861Q) |
ADP-Glo |
96/384 well |
EGFR(T790M,L858R) |
ADP-Glo |
96/384 well |
EGFR(T790M) |
ADP-Glo |
96/384 well |
EIF2AK2 |
ADP-Glo |
96/384 well |
EPHA1 |
ADP-Glo |
96/384 well |
ERK1 |
ADP-Glo |
96/384 well |
ERK2 |
ADP-Glo |
96/384 well |
FAK |
ADP-Glo |
96/384 well |
FES |
ADP-Glo |
96/384 well |
FGFR1 |
ADP-Glo |
96/384 well |
FGFR2 |
ADP-Glo |
96/384 well |
FGFR3(K650E) |
ADP-Glo |
96/384 well |
FGFR4 |
ADP-Glo |
96/384 well |
FLT1 |
ADP-Glo |
96/384 well |
FLT3 |
ADP-Glo |
96/384 well |
FLT3(D835Y) |
ADP-Glo |
96/384 well |
FMS |
ADP-Glo |
96/384 well |
FYN A |
ADP-Glo |
96/384 well |
GRK5 |
ADP-Glo |
96/384 well |
GSK3α |
ADP-Glo |
96/384 well |
GSK3β |
ADP-Glo |
96/384 well |
HER2 |
ADP-Glo |
96/384 well |
HER4 |
ADP-Glo |
96/384 well |
HIPK1 |
ADP-Glo |
96/384 well |
HPK1 | ADP-Glo | 96/384 well |
Target | Assay | Format |
IGF1R |
ADP-Glo |
96/384 well |
IKK |
ADP-Glo |
96/384 well |
IKKα |
ADP-Glo |
96/384 well |
InsR |
ADP-Glo |
96/384 well |
IRAK4 |
ADP-Glo |
96/384 well |
ITK |
ADP-Glo |
96/384 well |
JAK3 |
ADP-Glo |
96/384 well |
JNK1 |
ADP-Glo |
96/384 well |
JNK3 |
ADP-Glo |
96/384 well |
KDR |
ADP-Glo |
96/384 well |
KHS1 |
ADP-Glo |
96/384 well |
LCK |
ADP-Glo |
96/384 well |
Lipid kinase |
ADP-Glo |
96/384 well |
LRRK2 |
ADP-Glo |
96/384 well |
LYN B |
ADP-Glo |
96/384 well |
MAPKAPK2 |
ADP-Glo |
96/384 well |
MAPKAPK3 |
ADP-Glo |
96/384 well |
MAPKAPK5 |
ADP-Glo |
96/384 well |
MARK1 |
ADP-Glo |
96/384 well |
MELK |
ADP-Glo |
96/384 well |
MET |
ADP-Glo |
96/384 well |
MET(M1250T) |
ADP-Glo |
96/384 well |
MINK1 |
ADP-Glo |
96/384 well |
MLCK |
ADP-Glo |
96/384 well |
MLK1 |
ADP-Glo |
96/384 well |
MLK2 |
ADP-Glo |
96/384 well |
MRCKa |
ADP-Glo |
96/384 well |
MSK1 |
ADP-Glo |
96/384 well |
MSK2 |
ADP-Glo |
96/384 well |
MST1 |
ADP-Glo |
96/384 well |
MYO3β | ADP-Glo | 96/384 well |
Target | Assay | Format |
NEK2 |
ADP-Glo |
96/384 well |
NEK3 |
ADP-Glo |
96/384 well |
NIK |
ADP-Glo |
96/384 well |
NUAK2 |
ADP-Glo |
96/384 well |
p38α |
ADP-Glo |
96/384 well |
p38B |
ADP-Glo |
96/384 well |
p38γ |
ADP-Glo |
96/384 well |
P38δ |
ADP-Glo |
96/384 well |
p70S6K |
ADP-Glo |
96/384 well |
p70S6Kb |
ADP-Glo |
96/384 well |
PAK1/CDC42 |
ADP-Glo |
96/384 well |
PAK3 |
ADP-Glo |
96/384 well |
PAK4 |
ADP-Glo |
96/384 well |
PASK |
ADP-Glo |
96/384 well |
PDGFRa(D842V) |
ADP-Glo |
96/384 well |
PDGFRa(T674I) |
ADP-Glo |
96/384 well |
PDGFRα |
ADP-Glo |
96/384 well |
PDGFRβ |
ADP-Glo |
96/384 well |
PDK1 |
ADP-Glo |
96/384 well |
PI3K Lipid kinases |
ADP-Glo |
96/384 well |
PI3K-Glo |
ADP-Glo |
96/384 well |
PIM1 |
ADP-Glo |
96/384 well |
PIM2 |
ADP-Glo |
96/384 well |
PKA | ADP-Glo | 96/384 well |
Target | Assay | Format |
PKC |
ADP-Glo |
96/384 well |
PKC1 |
ADP-Glo |
96/384 well |
PKCα |
ADP-Glo |
96/384 well |
PKCβII |
ADP-Glo |
96/384 well |
PKCγ |
ADP-Glo |
96/384 well |
PKCδ |
ADP-Glo |
96/384 well |
PKCε |
ADP-Glo |
96/384 well |
PKCζ |
ADP-Glo |
96/384 well |
PKCθ |
ADP-Glo |
96/384 well |
PKCι |
ADP-Glo |
96/384 well |
PKCμ |
ADP-Glo |
96/384 well |
PKD2 |
ADP-Glo |
96/384 well |
PLK1 |
ADP-Glo |
96/384 well |
PRKG1 |
ADP-Glo |
96/384 well |
PYK2 |
ADP-Glo |
96/384 well |
RET |
ADP-Glo |
96/384 well |
RET(V804L) |
ADP-Glo |
96/384 well |
RET(Y791F) |
ADP-Glo |
96/384 well |
RIPK2 |
ADP-Glo |
96/384 well |
ROCK1 |
ADP-Glo |
96/384 well |
ROCK2 |
ADP-Glo |
96/384 well |
RON |
ADP-Glo |
96/384 well |
RSK1 |
ADP-Glo |
96/384 well |
SGK1 |
ADP-Glo |
96/384 well |
SIK |
ADP-Glo |
96/384 well |
SLK |
ADP-Glo |
96/384 well |
SRC |
ADP-Glo |
96/384 well |
STK33 |
ADP-Glo |
96/384 well |
SYK | ADP-Glo | 96/384 well |
Target | Assay | Format |
TAK1-TAB1 |
ADP-Glo |
96/384 well |
TAOK1 |
ADP-Glo |
96/384 well |
TBK1 |
ADP-Glo |
96/384 well |
TGFbR1 |
ADP-Glo |
96/384 well |
TGFβR2 |
ADP-Glo |
96/384 well |
TNIK |
ADP-Glo |
96/384 well |
TOPK |
ADP-Glo |
96/384 well |
TRKA |
ADP-Glo |
96/384 well |
TRKB |
ADP-Glo |
96/384 well |
ULK1 |
ADP-Glo |
96/384 well |
VRK2 |
ADP-Glo |
96/384 well |
WNK1 |
ADP-Glo |
96/384 well |
ZAK |
ADP-Glo |
96/384 well |
ZAP70 | ADP-Glo | 96/384 well |
激酶功能实验价格
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